SCHEMBL13543775

SCHEMBL13543775

Cc1nc2ccccc2n1[C@H]1C[C@H]2CC[C@@H](C1)N2CCC1(c2ccccc2)CCN(C(=O)c2ccc(Cl)c(N)c2)CC1

nearest known ligand 0.87

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 12/20 0.87
KCNH2 Q12809 10/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3528594 1.00 CCR5 (0.87) CCR5KCNH2
SCHEMBL13543409 0.93 CCR5 (1.00) CCR5KCNH2
SCHEMBL3530353 0.93 CCR5 (1.00) CCR5KCNH2
SCHEMBL13543816 0.90 CCR5 (0.89) CCR5KCNH2
SCHEMBL3529046 0.90 CCR5 (0.89) CCR5KCNH2
SCHEMBL3531169 0.90 CCR5 (0.83) CCR5KCNH2
SCHEMBL13543813 0.90 KCNH2 (0.87) CCR5KCNH2
SCHEMBL3531309 0.90 KCNH2 (0.87) CCR5KCNH2
SCHEMBL13543577 0.89 CCR5 (1.00) CCR5KCNH2
SCHEMBL13544043 0.89 CCR5 (1.00) CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed