SCHEMBL13544690

SCHEMBL13544690

CC(=O)c1cccc2[nH]c(C)nc12

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.73
DHODH Q02127 9/20 0.49
KDM4E B2RXH2 1/20 0.45
HPGD P15428 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1298127 0.86 PARP1 (0.73) PARP1DHODHKDM4EHPGD
SCHEMBL871829 0.85 PARP1 (1.00) PARP1DHODH
SCHEMBL7477535 0.82 PARP1 (0.68) PARP1DHODHKDM4E
SCHEMBL1193115 0.81 PARP1 (0.54) PARP1DHODHKDM4EHPGD
SCHEMBL14564598 0.81 PARP1 (0.50) PARP1DHODHKDM4EHPGD
SCHEMBL16555253 0.81 PARP1 (0.66) PARP1DHODHKDM4EHPGD
SCHEMBL6170661 0.80 PARP1 (0.64) PARP1DHODHKDM4E
SCHEMBL7333705 0.79 PARP1 (0.62) PARP1DHODHKDM4EHPGD
SCHEMBL17702653 0.78 L3MBTL1 (0.51) PARP1DHODHKDM4EHPGD
SCHEMBL23395014 0.77 DHODH (0.64) PARP1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed
US-7645771-B2 CCR5 antagonists as therapeutic agents SMITHKLINE BEECHAM CORP. (US) 2010-01-12 US disclosed