SCHEMBL13547660

SCHEMBL13547660

Bc1ccc(Nc2nc(Nc3ccc4[nH]ncc4c3)c3sccc3n2)nc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 9/20 0.51
ROCK1 Q13464 6/20 0.47
MKNK1 Q9BUB5 2/20 0.43
EGFR P00533 4/20 0.41
FLT1 P17948 3/20 0.41
RET P07949 2/20 0.41
CHEK1 O14757 1/20 0.41
AURKA O14965 1/20 0.41
DAPK3 O43293 1/20 0.41
JAK2 O60674 1/20 0.41
PRKD3 O94806 1/20 0.41
MAP4K4 O95819 1/20 0.41
PAK4 O96013 1/20 0.41
ABL1 P00519 1/20 0.41
NTRK1 P04629 1/20 0.41
LCK P06239 1/20 0.41
FYN P06241 1/20 0.41
CSF1R P07333 1/20 0.41
IGF1R P08069 1/20 0.41
MET P08581 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13547636 0.89 ROCK2 (0.55) ROCK2ROCK1MKNK1EGFRFLT1
SCHEMBL13220497 0.89 ROCK2 (0.51) ROCK2ROCK1MKNK1EGFRFLT1
SCHEMBL13220401 0.85 ROCK2 (0.52) ROCK2ROCK1MKNK1EGFRFLT1
SCHEMBL13220503 0.85 ROCK2 (0.51) ROCK2ROCK1MKNK1EGFRFLT1
SCHEMBL13547588 0.84 HSF1 (0.48) ROCK2ROCK1MKNK1EGFRFLT1
SCHEMBL13220518 0.84 ROCK2 (0.48) ROCK2ROCK1MKNK1EGFRFLT1
SCHEMBL13220333 0.83 ROCK2 (0.51) ROCK2ROCK1MKNK1EGFRFLT1
SCHEMBL13241612 0.81 ROCK2 (0.49) ROCK2ROCK1MKNK1EGFRFLT1
SCHEMBL13220452 0.81 ROCK2 (0.55) ROCK2ROCK1MKNK1EGFRFLT1
SCHEMBL13220422 0.81 ROCK2 (0.55) ROCK2ROCK1MKNK1EGFRFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7648986-B2 Substituted thieno[3,2-D]pyrimidines as Rho kinase inhibitors BAYER HEALTHCARE LLC (US) 2010-01-19 US disclosed