SCHEMBL13567643

SCHEMBL13567643

CCCCOc1ccc(COc2ccc(Br)cc2C(=N)C(=O)OC)cc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 9/20 0.47
AKR1C2 P52895 1/20 0.44
AKR1C1 Q04828 1/20 0.44
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
PDE4A P27815 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HIF1A Q16665 1/20 0.43
HDAC10 Q969S8 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
SMPD1 P17405 2/20 0.42
MAOB P27338 2/20 0.41
CCR5 P51681 2/20 0.41
MAOA P21397 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10049869 0.78 SMN1; SMN2 (0.48) KDM4ECYP1A2CYP2D6PDE4ASMN1; SMN2
SCHEMBL10050013 0.75 PTGER1 (0.48) KDM4ECYP1A2CYP2D6PDE4ASMN1; SMN2
SCHEMBL1646591 0.74 LRRK2 (0.61) LRRK2SMN1; SMN2SMPD1MAOBCCR5
SCHEMBL2772497 0.73 SMN1; SMN2 (0.49) AKR1C2AKR1C1KDM4ECYP1A2SMN1; SMN2
SCHEMBL548028 0.72 LRRK2 (0.53) LRRK2KDM4ECCR5
SCHEMBL6492975 0.72 LRRK2 (0.60) LRRK2KDM4EHDAC6SMPD1CCR5
SCHEMBL10049810 0.71 CNR2 (0.54) SMN1; SMN2CCR5
SCHEMBL13413498 0.71 MAPT (0.60) CYP1A2SMN1; SMN2HDAC6SMPD1
SCHEMBL1647292 0.71 LRRK2 (0.58) LRRK2KDM4ESMPD1MAOBCCR5
SCHEMBL16307018 0.70 PTGDR2 (0.66) AKR1C2AKR1C1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2128148-A1 COMPOUND, ALPHA 1 ADRENALINE RECEPTOR ANTAGONIST, AND COMPOSITION Suntory Holdings Limited (JP) 2009-12-02 EP disclosed