SCHEMBL1357023

SCHEMBL1357023

c1csc(-c2cncc(-c3cccs3)c2)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.67
CYP2E1 P05181 1/20 0.67
CYP3A4 P08684 1/20 0.67
CYP2C9 P11712 1/20 0.67
CYP2B6 P20813 1/20 0.67
CYP17A1 P05093 1/20 0.48
CYP11B1 P15538 1/20 0.48
CYP11B2 P19099 1/20 0.48
KCNH2 Q12809 1/20 0.48
PDGFRB P09619 1/20 0.46
PDGFRA P16234 1/20 0.46
KDM4E B2RXH2 4/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
HSD17B10 Q99714 2/20 0.46
RAB9A P51151 1/20 0.46
LTA4H P09960 1/20 0.45
ROCK1 Q13464 1/20 0.45
MAPT P10636 2/20 0.45
MEN1 O00255 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12608100 0.90 CYP2E1 (0.56) CYP2A6CYP2E1CYP3A4CYP2C9CYP2B6
SCHEMBL12608111 0.86 CYP2A6 (0.56) CYP2A6CYP2E1CYP3A4CYP2C9CYP2B6
SCHEMBL4135591 0.86 CYP2A6 (0.56) CYP2A6CYP2E1CYP3A4CYP2C9CYP2B6
SCHEMBL7423578 0.86 CYP3A4 (0.56) CYP2A6CYP2E1CYP3A4CYP2C9CYP2B6
SCHEMBL4135586 0.86 CYP2C9 (0.56) CYP2A6CYP2E1CYP3A4CYP2C9CYP2B6
SCHEMBL26387047 0.86 CYP2E1 (0.56) CYP2A6CYP2E1CYP3A4CYP2C9CYP2B6
SCHEMBL30613331 0.86 CYP2A6 (0.56) CYP2A6CYP2E1CYP3A4CYP2C9CYP2B6
SCHEMBL30722437 0.83 TOP1 (0.61) CYP2A6CYP2E1CYP3A4CYP2C9CYP2B6
SCHEMBL31418324 0.83 CYP3A4 (0.53) CYP2A6CYP2E1CYP3A4CYP2C9CYP2B6
SCHEMBL4338418 0.83 KCNH2 (0.58) CYP2A6CYP2E1CYP3A4CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9518964-B2 Method for identifying electrophiles and nucleophiles in a sample EICHEN YOAV (IL) 2016-12-13 US disclosed
US-9518964-B2 Method for identifying electrophiles and nucleophiles in a sample EICHEN YOAV (IL) 2016-12-13 US disclosed
US-9518964-B2 Method for identifying electrophiles and nucleophiles in a sample EICHEN YOAV (IL) 2016-12-13 US disclosed
US-20110281742-A1 METHOD FOR IDENTIFYING ELECTROPHILES AND NUCLEOPHILES IN A SAMPLE EICHEN YOAV (IL) 2011-11-17 US disclosed
US-20110281742-A1 METHOD FOR IDENTIFYING ELECTROPHILES AND NUCLEOPHILES IN A SAMPLE EICHEN YOAV (IL) 2011-11-17 US disclosed
US-20110281742-A1 METHOD FOR IDENTIFYING ELECTROPHILES AND NUCLEOPHILES IN A SAMPLE EICHEN YOAV (IL) 2011-11-17 US disclosed
US-20090258430-A1 Method for identifying electrophiles and nucleophiles in a sample TECHNION RESEARCH & DEVELOPMENT FOUNDATION LTD. (IL) 2009-10-15 US disclosed
US-20090258430-A1 Method for identifying electrophiles and nucleophiles in a sample TECHNION RESEARCH & DEVELOPMENT FOUNDATION LTD. (IL) 2009-10-15 US disclosed
US-20090258430-A1 Method for identifying electrophiles and nucleophiles in a sample TECHNION RESEARCH & DEVELOPMENT FOUNDATION LTD. (IL) 2009-10-15 US disclosed
EP-2085766-A2 Method for identifying electrophiles and nucleophiles in a sample Technion Research and Development Foundation, Ltd. (IL) 2009-08-05 EP disclosed
EP-2085766-A2 Method for identifying electrophiles and nucleophiles in a sample Technion Research and Development Foundation, Ltd. (IL) 2009-08-05 EP disclosed