SCHEMBL13574641

SCHEMBL13574641

c1ccc(CNc2nccc(N3CCCC3)n2)nc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OGA O60502 5/20 0.61
CXCR4 P61073 2/20 0.60
ADORA2A P29274 1/20 0.56
ADORA1 P30542 1/20 0.56
HRH4 Q9H3N8 8/20 0.50
HRH3 Q9Y5N1 3/20 0.50
ADRA2B P18089 2/20 0.50
ADRA2C P18825 2/20 0.50
SLC6A2 P23975 2/20 0.50
HTR1D P28221 2/20 0.50
HTR2C P28335 2/20 0.50
HTR2B P41595 2/20 0.50
HRH2 P25021 1/20 0.50
HTR2A P28223 1/20 0.50
HTR7 P34969 1/20 0.50
HTR5A P47898 1/20 0.50
HTR6 P50406 1/20 0.50
SLC6A3 Q01959 1/20 0.50
TMEM97 Q5BJF2 1/20 0.50
SIGMAR1 Q99720 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1088599 0.99 CXCR4 (0.63) OGACXCR4ADORA2AADORA1HRH4
SCHEMBL1588315 0.88 HRH4 (0.63) OGACXCR4HRH4HRH3ADRA2B
SCHEMBL1587997 0.88 HRH4 (0.66) OGACXCR4HRH4HRH3ADRA2B
SCHEMBL26708280 0.83 CXCR4 (0.63) OGACXCR4HRH4HRH3ADRA2B
SCHEMBL847331 0.81 HRH4 (0.65) OGAHRH4HRH3ADRA2BADRA2C
SCHEMBL1589282 0.81 HRH4 (0.65) OGAHRH4HRH3ADRA2BADRA2C
SCHEMBL19459031 0.81 HRH4 (0.65) OGAHRH4HRH3ADRA2BADRA2C
SCHEMBL847664 0.81 OGA (0.56) OGAHRH4HRH3ADRA2BADRA2C
SCHEMBL1822887 0.80 HRH4 (0.67) OGAHRH4HRH3ADRA2BADRA2C
SCHEMBL860555 0.80 OGA (0.60) OGAHRH4HRH3ADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009152325-A1 DIAMINO-PYRIDINE, PYRIMIDINE, AND PYRIDAZINE MODULATORS OF THE HISTAMINE H4 RECEPTOR JANSSEN PHARMACEUTICA NV (BE) 2009-12-17 WO disclosed