SCHEMBL13577960

SCHEMBL13577960

COC(=O)c1ccc2c(C3CCCCC3)cn(CCCCN)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 0.46
SCN5A Q14524 2/20 0.46
CNR2 P34972 3/20 0.43
CNR1 P21554 1/20 0.43
ALDH1A1 P00352 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
HPGD P15428 1/20 0.42
CYP2C19 P33261 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
PDE4A P27815 3/20 0.40
PDE4B Q07343 3/20 0.40
PDE4C Q08493 3/20 0.40
PDE4D Q08499 3/20 0.40
PRPS1 P60891 2/20 0.39
TLR8 Q9NR97 2/20 0.39
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4827022 0.89 SCN9A (0.46) SCN9ASCN5ACNR2CNR1ALDH1A1
SCHEMBL4830054 0.87 SCN9A (0.49) SCN9ASCN5ACNR2CNR1ALDH1A1
SCHEMBL13577940 0.85 HPGD (0.44) SCN9ASCN5ACNR2CNR1ALDH1A1
SCHEMBL14435340 0.84 SCN9A (0.45) SCN9ASCN5ACNR2CNR1ALDH1A1
SCHEMBL772052 0.82 HRH2 (0.44) SCN9ASCN5ACNR2CNR1ALDH1A1
SCHEMBL13577944 0.82 LMNA (0.45) SCN9ASCN5ACNR2CNR1ALDH1A1
SCHEMBL1260945 0.81 SCN9A (0.65) SCN9ASCN5ACNR2CNR1ALDH1A1
SCHEMBL899454 0.80 SCN9A (0.64) SCN9ASCN5ACNR2CNR1ALDH1A1
SCHEMBL4831650 0.80 HRH2 (0.48) SCN9ASCN5ACNR2HRH2
SCHEMBL4324275 0.79 TLR8 (0.43) CNR2CNR1ALDH1A1KDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009147121-A1 CARBOXYL SUBSTITUTED INDOLES FOR USE AS PPAR ALPHA MODULATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-12-10 WO disclosed