SCHEMBL1358362

SCHEMBL1358362

CC(C)(C)c1cc(-c2ccc[nH]c2=O)cc2c(-c3cccc(CNS(C)(=O)=O)c3)coc12

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.44
BRD4 O60885 3/20 0.42
CREBBP Q92793 2/20 0.41
IGLV6-57 P01721 1/20 0.35
IGF1R P08069 1/20 0.34
MET P08581 1/20 0.34
SRC P12931 1/20 0.34
AAK1 Q2M2I8 1/20 0.33
AURKA O14965 2/20 0.32
AURKB Q96GD4 2/20 0.32
NFATC1 O95644 1/20 0.32
CSNK1D P48730 1/20 0.32
CSNK1E P49674 1/20 0.32
LIPG Q9Y5X9 1/20 0.31
IKBKB O14920 1/20 0.30
CHUK O15111 1/20 0.30
PDCD1 Q15116 1/20 0.30
CD274 Q9NZQ7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1358298 0.91 CYP3A4 (0.47) CYP3A4BRD4CREBBP
SCHEMBL1360136 0.85 CYP3A4 (0.38) CYP3A4IGLV6-57
SCHEMBL1359875 0.85 CYP3A4 (0.49) CYP3A4BRD4CREBBP
SCHEMBL1359885 0.84 NFATC1 (0.45) CYP3A4BRD4CREBBPIGF1RMET
SCHEMBL1359216 0.84 CYP3A4 (0.47) CYP3A4
SCHEMBL1359902 0.84 CYP3A4 (0.40) CYP3A4
SCHEMBL1358305 0.81 CYP3A4 (0.55) CYP3A4IKBKBCHUK
SCHEMBL1358251 0.81 CYP3A4 (0.38) CYP3A4
SCHEMBL1359548 0.80 BRAF (0.36) CYP3A4
SCHEMBL1358345 0.80 CYP3A4 (0.41) CYP3A4CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8067442-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2011-11-29 US claimed
US-20100081658-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS ROCHE PALO ALTO LLC 2010-04-01 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100081658-A1 HETEROCYCLIC ANTIVIRAL COMPOUNDS EIF2AK2, POLR2A, HCCS CYP3A4 713/4885BRD4 1086/4885CREBBP 1002/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.