SCHEMBL13595347

SCHEMBL13595347

COC(=O)c1c(-c2ccc(O)cc2)c(-c2ccc(O)cc2)cn1CC(=O)c1ccc(O)cc1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.38
CA1 P00915 4/20 0.38
CA2 P00918 4/20 0.38
CA7 P43166 4/20 0.38
CA9 Q16790 4/20 0.38
CA14 Q9ULX7 4/20 0.38
PDK2 Q15119 1/20 0.38
PDK4 Q16654 1/20 0.38
HSD17B1 P14061 1/20 0.38
TP53 P04637 2/20 0.37
NPC1 O15118 1/20 0.37
MAPK1 P28482 1/20 0.37
EGFR P00533 1/20 0.35
HPGD P15428 3/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HSD17B10 Q99714 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5820726 0.81 ESR2 (0.47) CA1CA2NPC1ALDH1A1KDM4E
SCHEMBL5775199 0.81 ESR2 (0.47) CA1CA2NPC1ALDH1A1KDM4E
SCHEMBL5946174 0.71 CA12 (0.44) CA12CA1CA2CA7CA9
SCHEMBL5946082 0.70 CYP1A2 (0.42) EGFRHPGDMEN1KMT2AALDH1A1
SCHEMBL13595362 0.69 ESRRA (0.45) CA12CA1CA2CA7CA9
SCHEMBL131661 0.69 CA12 (0.69) CA12CA1CA2CA7CA9
SCHEMBL2770758 0.68 HSD17B1 (0.56) CA12CA1CA2CA7CA9
SCHEMBL497983 0.67 HSD17B1 (0.69) CA12CA1CA2CA7CA9
SCHEMBL28675075 0.66 CA12 (0.56) CA12CA1CA2CA7CA9
SCHEMBL27735150 0.66 HSP90AB1 (0.53) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2138496-A1 Antitumoral analogs of lamellarins Pharma Mar, S.A.U. (ES) 2009-12-30 EP disclosed
US-7396837-B2 Antitumoral analogs of lamellarins PHARMA MAR, S.A.U. (ES) 2008-07-08 US disclosed