SCHEMBL13601359

SCHEMBL13601359

C1=C(c2cccc(-c3nnn[nH]3)c2)c2ccccc2OC12CCNCC2

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 20/20 0.63
KCNH2 Q12809 16/20 0.63
OPRK1 P41145 6/20 0.63
CYP2D6 P10635 11/20 0.51
OPRM1 P35372 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL471286 0.81 OPRD1 (0.63) OPRD1KCNH2OPRK1CYP2D6OPRM1
SCHEMBL467151 0.79 OPRD1 (1.00) OPRD1KCNH2OPRK1CYP2D6OPRM1
SCHEMBL471263 0.78 OPRD1 (0.75) OPRD1KCNH2OPRK1CYP2D6OPRM1
SCHEMBL471270 0.78 OPRD1 (0.60) OPRD1KCNH2OPRK1CYP2D6OPRM1
Hydrochloric Acid SCHEMBL12481185 0.78 OPRD1 (0.97) OPRD1KCNH2OPRK1CYP2D6OPRM1
SCHEMBL10259459 0.77 OPRD1 (0.76) OPRD1KCNH2OPRK1CYP2D6OPRM1
SCHEMBL10257844 0.76 OPRD1 (0.60) OPRD1KCNH2OPRK1CYP2D6OPRM1
SCHEMBL471272 0.76 OPRD1 (0.77) OPRD1KCNH2OPRK1CYP2D6OPRM1
SCHEMBL471265 0.74 OPRD1 (0.74) OPRD1KCNH2OPRK1CYP2D6OPRM1
SCHEMBL10258871 0.73 OPRD1 (0.73) OPRD1KCNH2OPRK1CYP2D6OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7638527-B2 Spirocyclic heterocyclic derivatives and methods of their use ADOLOR CORPORATION (US) 2009-12-29 US disclosed
US-7638527-B2 Spirocyclic heterocyclic derivatives and methods of their use ADOLOR CORPORATION (US) 2009-12-29 US disclosed