SCHEMBL1360313

SCHEMBL1360313

C[C@H](NC(=O)Cc1cc(F)cc(F)c1)C(=O)N[C@H](C(=O)OC(C)(C)C)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 14/20 0.47
PSEN2 P49810 14/20 0.47
APH1B Q8WW43 14/20 0.47
NCSTN Q92542 14/20 0.47
APH1A Q96BI3 14/20 0.47
PSENEN Q9NZ42 14/20 0.47
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
GSAP A4D1B5 1/20 0.43
REN P00797 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CNR2 P34972 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14876684 1.00 PSEN1 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL23476580 1.00 PSEN1 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL1360317 1.00 PSEN1 (0.47) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL14886930 0.89 CYP3A4 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL18642504 0.86 CYP3A4 (0.51) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL28186177 0.86 CYP3A4 (0.51) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5966881 0.84 KLK5 (0.48) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL16490908 0.84 PSEN1 (0.45) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL5967121 0.84 REN (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4057116 0.84 PSEN1 (0.42) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2845 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4747363-A1 NEURAL DIFFERENTIATION FROM PLURIPOTENT CELLS Treefrog Therapeutics (FR) 2026-05-27 EP claimed
CN-121526349-B Dynamic risk management method and system for traffic engineering construction XIAMEN ROAD & BRIDGE INFORMATION Co.,Ltd. (CN) 2026-05-26 CN claimed
US-12629337-B2 Daptomycin formulation HIKMA PHARMACEUTICALS USA INC. (US) 2026-05-19 US claimed
US-20260132374-A1 Compositions and Methods for Efficient Amplification of Retinal Progenitors Cells SORBONNE UNIVERSITE (FR) 2026-05-14 US claimed
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES TRAILHEAD BIOSYSTEMS INC (US) 2026-05-07 US claimed
US-12618044-B2 Specification of functional cranial placode derivatives from human pluripotent stem cells MEMORIAL SLOAN-KETTERING CANCER CENTER (US) 2026-05-05 US claimed
WO-2026089437-A1 LIVER TISSUE-LIKE ORGANOID AND METHOD OF MANUFACTURING THE SAME KOREA RESEARCH INSTITUTE OF BIOSCIENCE AND BIOTECHNOLOGY (KR) 2026-04-30 WO claimed
WO-2026088216-A1 METHOD OF GENERATING LIVER ORGANOID MODEL AND MODEL RECAPITULATING NAFLD HALLMARKS TRANSLATIONAL HEALTH SCIENCE AND TECHNOLOGY INSTITUTE (IN) 2026-04-30 WO claimed
US-20260117188-A1 LIVER TISSUE-LIKE ORGANOID AND METHOD OF MANUFACTURING THE SAME KOREA RES INST BIOSCIENCE & BIOTECHNOLOGY (KR) 2026-04-30 US claimed
EP-4720261-A1 NOVEL CULTURE CONDITIONS FOR CLONAL EXPANSION OF NEPHRON PROGENITOR CELLS, GENERATION OF NEPHRON ORGANOIDS, AND RAPID AND SCALABLE MODELING OF POLYCYSTIC KIDNEY DISEASE University of Southern California (US) 2026-04-08 EP claimed
US-20220062291-A1 COMPOSITIONS AND METHODS OF TREATING CANCERS BY ADMINISTERING A PHENOTHIAZINE-RELATED DRUG THAT ACTIVATES PROTEIN PHOSPHATASE 2A (PP2A) WITH REDUCED INHIBITORY ACTIVITY TARGETED TO THE DOPAMINE D2 RECEPTOR AND ACCOMPANYING TOXICITY DANA-FARBER CANCER INSTITUTE, INC. (US) 2022-03-03 US claimed
EP-3959306-A1 NOCICEPTOR DIFFERENTIATION FROM HUMAN PLURIPOTENT STEM CELLS The United States of America as represented by the Secretary of the Department of Health and Human Services (US) 2022-03-02 EP claimed
CN-114096557-A Generation of germ layer cells in the dorsal foregut and anterior structural domains 克利夫兰诊所基金会 2022-02-25 CN claimed
EP-3303564-B1 METHODS OF IN VITRO DIFFERENTIATION OF MIDBRAIN DOPAMINE (MDA) NEURONS MEMORIAL SLOAN KETTERING CANCER CENTER (US) 2022-02-23 EP claimed
US-11254916-B2 Methods of making and using PDX1-positive pancreatic endoderm cells VIACYTE, INC. (US) 2022-02-22 US claimed
CN-111500526-B Composition for in-vitro culture of primary mouse corneal epithelial cells and application thereof 厦门大学 2022-02-18 CN claimed
US-20220041990-A1 METHODS, COMPOSITIONS, AND KITS FOR PRODUCING SKELETAL MUSCLE STEM CELLS AND TREATING DISORDERS UNIV JOHNS HOPKINS (US) 2022-02-10 US claimed
EP-3945827-A2 METHODS, COMPOSITIONS, AND KITS FOR PRODUCING SKELETAL MUSCLE STEM CELLS AND TREATING DISORDERS The Johns Hopkins University (US) 2022-02-09 EP claimed
WO-2022026932-A2 DIFFERENTIATION OF PANCREATIC ENDOCRINE CELLS VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-02-03 WO claimed
CN-110582564-A derivation of liver organoids from human pluripotent stem cells 新加坡科技研究局 2019-12-17 CN claimed