SCHEMBL13607828

SCHEMBL13607828

COc1ccc(Cc2nc3cc(Br)cnc3[nH]2)cc1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.47
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.41
RNASEH1 O60930 1/20 0.40
NQO2 P16083 3/20 0.39
CCNB2 O95067 1/20 0.39
CCNE2 O96020 1/20 0.39
CDK1 P06493 1/20 0.39
CCNB1 P14635 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
CCNB3 Q8WWL7 1/20 0.39
PDGFRB P09619 1/20 0.36
PDGFRA P16234 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13607783 0.92 POLB (0.57) POLBKDM4EALDH1A1GAAHPGD
SCHEMBL13607772 0.84 GRIN1 (0.47) POLBGAAPDGFRBSMN1; SMN2GRIN1
SCHEMBL13607808 0.83 ALDH1A1 (0.42) POLBALDH1A1GAACCNB2CDK1
SCHEMBL13608262 0.83 POLB (0.50) POLBKDM4EALDH1A1HPGDPDGFRB
SCHEMBL13607781 0.81 SMN1; SMN2 (0.48) POLBALDH1A1SMN1; SMN2GRIN1GRIN2B
SCHEMBL13607812 0.81 POLB (0.44) POLBKDM4EGAASMN1; SMN2
SCHEMBL4058869 0.81 RXFP1 (0.54) POLBKDM4EALDH1A1GAAHPGD
SCHEMBL13607799 0.81 CDK5 (0.48) POLBALDH1A1GAACCNB2CDK1
SCHEMBL13607782 0.80 HSP90AA1 (0.47) POLBPDGFRBSMN1; SMN2DHFRHTT
SCHEMBL13608281 0.79 POLB (0.43) POLBKDM4EALDH1A1GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622479-B2 Bicyclic derivative, its production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed
US-7622479-B2 Bicyclic derivative, its production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed