SCHEMBL13610549

SCHEMBL13610549

COc1ccc2c(c1)CCN=C2CCl

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.60
KDM4E B2RXH2 3/20 0.60
LMNA P02545 2/20 0.60
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
MPO P05164 1/20 0.48
CYP1A2 P05177 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
HSD17B10 Q99714 1/20 0.44
GLA P06280 1/20 0.44
RCE1 Q9Y256 1/20 0.44
CYP19A1 P11511 5/20 0.43
CYP11B2 P19099 4/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL329858 0.98 ALDH1A1 (0.62) ALDH1A1KDM4ELMNACA1CA2
Hydrochloric Acid SCHEMBL3450797 0.88 KDM4E (0.51) ALDH1A1KDM4ELMNACA1CA2
SCHEMBL18183525 0.87 ALDH1A1 (0.63) ALDH1A1KDM4ELMNACA1CA2
SCHEMBL13869188 0.84 ALDH1A1 (0.60) ALDH1A1KDM4ELMNACA1CA2
SCHEMBL24528920 0.83 KDM4E (0.59) ALDH1A1KDM4ELMNACA1CA2
Hydrochloric Acid SCHEMBL330055 0.83 ALDH1A1 (0.62) ALDH1A1KDM4ELMNACA1CA2
SCHEMBL17144585 0.80 CA1 (0.66) ALDH1A1KDM4ELMNACA1CA2
SCHEMBL21346192 0.80 KDM4E (0.73) ALDH1A1KDM4ELMNACA1CA2
SCHEMBL10961422 0.80 KDM4E (0.69) ALDH1A1KDM4ELMNACA1CA2
SCHEMBL10737635 0.79 CYP1A2 (0.68) ALDH1A1KDM4ELMNACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090286843-A1 MACROCYCLIC COMPOUNDS AS INHIBITORS OF VIRAL REPLICATION HOFFMANN-LA ROCHE INC. 2009-11-19 US disclosed
US-20090111969-A1 MACROCYCLIC COMPOUNDS AS INHIBITORS OF VIRAL REPLICATION HOFFMANN-LA ROCHE INC. 2009-04-30 US disclosed
US-20090111982-A1 MACROCYCLIC COMPOUNDS AS INHIBITORS OF VIRAL REPLICATION HOFFMANN-LA ROCHE INC. 2009-04-30 US disclosed
US-20090105471-A1 MACROCYCLIC COMPOUNDS AS INHIBITORS OF VIRAL REPLICATION HOFFMANN-LA ROCHE INC. 2009-04-23 US disclosed
US-7491794-B2 Macrocyclic compounds as inhibitors of viral replication INTERMUNE, INC. (US) 2009-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090111982-A1 MACROCYCLIC COMPOUNDS AS INHIBITORS OF VIRAL REPLICATION EIF2AK2, HAVCR2, ZC3HAV1 ALDH1A1 2109/4885KDM4E 616/4885LMNA 625/4885
US-20090286843-A1 MACROCYCLIC COMPOUNDS AS INHIBITORS OF VIRAL REPLICATION EIF2AK2, HAVCR2, ZC3HAV1 ALDH1A1 2109/4885KDM4E 616/4885LMNA 625/4885
US-20090111969-A1 MACROCYCLIC COMPOUNDS AS INHIBITORS OF VIRAL REPLICATION EIF2AK2, HAVCR2, ZC3HAV1 ALDH1A1 2109/4885KDM4E 616/4885LMNA 625/4885
US-20090105471-A1 MACROCYCLIC COMPOUNDS AS INHIBITORS OF VIRAL REPLICATION EIF2AK2, HAVCR2, ZC3HAV1 ALDH1A1 2109/4885KDM4E 616/4885LMNA 625/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.