SCHEMBL13617396

SCHEMBL13617396

CCCCOc1ccc([C@@H](O)CNCCc2ccc(Nc3ccc(S(=O)(=O)Nc4ccccn4)cc3)cc2)c2ccc(=O)[nH]c12

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 20/20 0.55
ADRB1 P08588 16/20 0.53
ADRB3 P13945 15/20 0.53
DRD2 P14416 2/20 0.52
DRD1 P21728 2/20 0.52
DRD4 P21917 2/20 0.52
DRD3 P35462 2/20 0.52
CHRM2 P08172 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13617478 0.87 ADRB2 (0.64) ADRB2ADRB1ADRB3CHRM2
SCHEMBL13617623 0.83 ADRB2 (0.78) ADRB2ADRB1ADRB3DRD2DRD1
SCHEMBL13589488 0.81 ADRB2 (0.80) ADRB2ADRB1ADRB3DRD2DRD1
SCHEMBL13711797 0.80 ADRB2 (0.62) ADRB2ADRB1ADRB3DRD2DRD1
SCHEMBL13617404 0.80 ADRB2 (0.61) ADRB2ADRB1ADRB3DRD2DRD1
SCHEMBL13711791 0.79 ADRB2 (0.69) ADRB2ADRB1ADRB3DRD2DRD1
SCHEMBL13617642 0.79 ADRB2 (0.52) ADRB2ADRB1ADRB3
SCHEMBL13617485 0.78 ADRB2 (0.59) ADRB2ADRB1ADRB3DRD2DRD1
SCHEMBL13617660 0.78 ADRB2 (0.54) ADRB2ADRB1ADRB3DRD2DRD1
SCHEMBL13708434 0.77 ADRB2 (0.40) ADRB2ADRB1ADRB3DRD2DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1641465-B1 COMBINATIONS OF AN ARYL ANILINE BETA-2 ADRENERGIC RECEPTOR AGONIST AND A CORTICOSTEROID THERAVANCE INC (US) 2009-11-04 EP disclosed
EP-1446379-B1 ARYL ANILINE BETA-2 ADRENERGIC RECEPTOR AGONISTS THERAVANCE INC (US) 2009-04-29 EP disclosed