SCHEMBL13617692

SCHEMBL13617692

CC(C)Cc1ccc(OCCCn2ccnn2)cc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 1/20 0.50
ATP4B P51164 1/20 0.50
CYP19A1 P11511 4/20 0.45
QPCT Q16769 1/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
ATM Q13315 1/20 0.37
ERBB2 P04626 1/20 0.37
MINK1 Q8N4C8 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
ACACB O00763 1/20 0.36
POLB P06746 1/20 0.36
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA9 Q16790 1/20 0.35
PDGFRB P09619 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14996228 0.85 ATP4A (0.53) ATP4AATP4BCYP19A1QPCTMEN1
SCHEMBL22397927 0.81 MEN1 (0.55) ATP4AATP4BCYP19A1QPCTMEN1
SCHEMBL765017 0.81 QPCT (0.56) ATP4AATP4BCYP19A1QPCTMEN1
SCHEMBL13201562 0.81 ATP4A (0.53) ATP4AATP4BCYP19A1ERBB2MINK1
SCHEMBL14189706 0.79 ATP4A (0.52) ATP4AATP4BCYP19A1MEN1KMT2A
SCHEMBL5564341 0.79 ATP4A (0.52) ATP4AATP4BCYP19A1QPCTMEN1
SCHEMBL5046643 0.79 ATP4A (0.52) ATP4AATP4BCYP19A1QPCTMEN1
SCHEMBL18837867 0.79 ATP4A (0.52) ATP4AATP4BCYP19A1QPCTMEN1
SCHEMBL13617693 0.79 CYP3A4 (0.43) CYP19A1QPCTMEN1KMT2AATM
SCHEMBL16417747 0.78 MEN1 (0.59) ATP4AATP4BCYP19A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8455497-B2 Inhibitors of aspartyl protease VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-06-04 US disclosed
US-20090274650-A1 INHIBITORS OF ASPARTYL PROTEASE VERTEX PHARMACEUTICALS INCORPORATED 2009-11-05 US disclosed
US-20090274650-A1 INHIBITORS OF ASPARTYL PROTEASE VERTEX PHARMACEUTICALS INCORPORATED 2009-11-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090274650-A1 INHIBITORS OF ASPARTYL PROTEASE SPINT2, DNPEP, PRSS1 ATP4A 1393/4885ATP4B 1730/4885CYP19A1 2353/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.