SCHEMBL13619474

SCHEMBL13619474

CCc1ccccc1NC(=O)CSC(=O)NNC(=O)[C@H](CCSC)NC(=O)OC(C)(C)C

nearest known ligand 0.76

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSL P07711 7/20 0.76
ALDH1A1 P00352 4/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
TSHR P16473 3/20 0.48
KLK5 Q9Y337 1/20 0.45
CTSS P25774 2/20 0.45
CTSK P43235 2/20 0.45
KLK7 P49862 1/20 0.43
CA2 P00918 1/20 0.43
KDM4E B2RXH2 2/20 0.41
MAPT P10636 1/20 0.41
REN P00797 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12371560 0.90 CTSL (0.80) CTSLALDH1A1SMN1; SMN2TSHRCTSS
SCHEMBL12371605 0.87 CTSL (0.79) CTSLALDH1A1SMN1; SMN2TSHRCTSS
SCHEMBL12370616 0.87 CTSL (0.62) CTSLALDH1A1SMN1; SMN2TSHRKLK5
SCHEMBL12371441 0.85 CTSL (0.75) CTSLALDH1A1SMN1; SMN2TSHR
SCHEMBL12370596 0.83 CTSL (0.73) CTSLALDH1A1SMN1; SMN2TSHRKLK5
SCHEMBL12371564 0.83 CTSL (0.73) CTSLALDH1A1SMN1; SMN2TSHRKLK5
SCHEMBL12370593 0.83 CTSL (0.73) CTSLALDH1A1SMN1; SMN2TSHRCTSS
SCHEMBL12370563 0.81 CTSL (0.73) CTSLALDH1A1SMN1; SMN2TSHRCTSS
SCHEMBL30257292 0.81 CTSL (1.00) CTSLSMN1; SMN2KLK5CTSSCTSK
SCHEMBL12370557 0.81 CTSL (0.81) CTSLALDH1A1SMN1; SMN2TSHRCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009136997-A2 INHIBITORS OF HUMAN CATHEPSIN L, CATHEPSIN B, AND CATHEPSIN S THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2009-11-12 WO disclosed