SCHEMBL13620320

SCHEMBL13620320

COc1cccc(-c2ccc3nc(-c4cccc(N)c4)oc3c2)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 10/20 0.64
RAB9A P51151 10/20 0.64
KDM4E B2RXH2 8/20 0.64
SMN1; SMN2 Q16637 7/20 0.64
ALDH1A1 P00352 7/20 0.64
HPGD P15428 7/20 0.64
MAPT P10636 6/20 0.64
LMNA P02545 1/20 0.61
CASP3 P42574 1/20 0.61
NFKB1 P19838 2/20 0.58
NFKB2 Q00653 2/20 0.58
RELA Q04206 2/20 0.58
GLA P06280 2/20 0.58
HSD17B10 Q99714 2/20 0.58
TP53 P04637 2/20 0.58
TDP1 Q9NUW8 2/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
GPR119 Q8TDV5 2/20 0.56
KMT2A Q03164 8/20 0.52
MEN1 O00255 4/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4052772 0.92 NPC1 (0.69) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL4059683 0.88 NPC1 (0.65) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL4056991 0.87 NPC1 (0.62) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL4052671 0.87 NPC1 (0.62) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL4053396 0.86 RAB9A (0.70) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL4052771 0.85 NPC1 (0.61) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL13620435 0.85 HSD17B10 (0.62) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL4053485 0.85 NPC1 (0.66) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL2245027 0.83 RAB9A (0.69) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL4055495 0.83 NPC1 (0.58) NPC1RAB9AKDM4ESMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622479-B2 Bicyclic derivative, its production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed