Cocaine

Cocaine

SCHEMBL13624557

COC(=O)[C@@H]1C2CC[C@H](C[C@@H]1OC(=O)c1ccccc1)N2C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9A

The experimentally established mechanism targets of Cocaine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCN1A known ✓ P35498 1/20 1.00
SCN2A known ✓ Q99250 1/20 1.00
SCN3A known ✓ Q9NY46 1/20 1.00
KCNH2 Q12809 2/20 1.00
SLC6A2 P23975 2/20 1.00
SLC6A4 P31645 2/20 1.00
SLC6A3 Q01959 2/20 1.00
MAPT P10636 1/20 1.00
MAOA P21397 1/20 1.00
SIGMAR1 Q99720 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cocaine SCHEMBL26609 1.00 KCNH2 (1.00) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Cocaine SCHEMBL8440314 1.00 KCNH2 (1.00) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Cocaine SCHEMBL21931 1.00 KCNH2 (1.00) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Cocaine SCHEMBL16922143 1.00 KCNH2 (1.00) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Cocaine SCHEMBL5991910 1.00 KCNH2 (1.00) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Cocaine SCHEMBL23086019 1.00 KCNH2 (1.00) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Cocaine SCHEMBL20390951 1.00 KCNH2 (1.00) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Cocaine SCHEMBL10066803 1.00 KCNH2 (1.00) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Cocaine SCHEMBL21189582 1.00 KCNH2 (1.00) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Cocaine SCHEMBL21930 1.00 KCNH2 (1.00) KCNH2SLC6A2SLC6A4SLC6A3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009141627-A1 TREATING NIEMANN-PICK DISEASE TYPE C AND RELATED DISORDERS BY ELEVATING INTRACELLULAR CALCIUM ISIS INNOVATION LIMITED (GB) 2009-11-26 WO disclosed