SCHEMBL13624607

SCHEMBL13624607

C=C1CC[C@H](c2ccccc2)N1C(=O)[C@H](CC[C@H](O[Si](C)(C)C)c1ccc(F)cc1)[C@H](Nc1ccc(F)cc1)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37
ALDH1A1 P00352 4/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
RECQL P46063 1/20 0.34
PRKAA2 P54646 1/20 0.33
CHRM4 P08173 1/20 0.33
MAPT P10636 2/20 0.33
RAB9A P51151 2/20 0.33
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
AR P10275 1/20 0.33
LMNA P02545 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ACACB O00763 1/20 0.33
S1PR5 Q9H228 1/20 0.33
FFAR1 O14842 1/20 0.33
YAP1 P46937 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL524752 0.80 GRIN1 (0.37) GRIN1GRIN2BALDH1A1MEN1KMT2A
SCHEMBL3912213 0.79 IDH1 (0.34) ALDH1A1SMN1; SMN2
SCHEMBL10045761 0.79 IDH1 (0.34) ALDH1A1SMN1; SMN2
SCHEMBL13412438 0.79 IDH1 (0.34) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL12973889 0.78 IDH1 (0.33) ALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL12973852 0.78 IDH1 (0.34) ALDH1A1SMN1; SMN2
SCHEMBL12973868 0.77 IDH1 (0.36) ALDH1A1SMN1; SMN2
SCHEMBL5737415 0.77 IDH1 (0.33)
SCHEMBL13930594 0.76 ALDH1A1 (0.36) GRIN1GRIN2BALDH1A1MEN1KMT2A
SCHEMBL12973946 0.76 IDH1 (0.33) ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009140932-A2 METHOD OF PRODUCING (3R,4S)-L-(4-FLUOROPHENYL)-3-[(3S)-3-(4-FLUOROPHENYL)- HYDROXYPROPYL)]-4-(4-HYDROXYPHENYL)-2-AZETIDINONE ZENTIVA, K.S. (CZ) 2009-11-26 WO disclosed