SCHEMBL13625563

SCHEMBL13625563

O=C([C@@H]1CCCNC1)N(Cc1cc(Br)cc(Cl)c1Cl)C1CC1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 9/20 0.51
SLC6A2 P23975 8/20 0.51
SLC6A3 Q01959 3/20 0.47
REN P00797 11/20 0.46
KCNH2 Q12809 8/20 0.44
CYP3A4 P08684 3/20 0.43
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13625719 0.81 REN (0.60) RENKCNH2CYP3A4
SCHEMBL663581 0.81 SLC6A4 (0.44) SLC6A4SLC6A2SLC6A3RENKCNH2
SCHEMBL24872977 0.79 REN (0.57) SLC6A4SLC6A2SLC6A3RENKCNH2
SCHEMBL31258379 0.78 REN (0.58) SLC6A4SLC6A2SLC6A3RENKCNH2
SCHEMBL13625716 0.76 REN (0.58) RENKCNH2CYP3A4
SCHEMBL13625723 0.74 REN (0.58) SLC6A4SLC6A2RENKCNH2CYP3A4
SCHEMBL13617898 0.72 REN (0.54) SLC6A4SLC6A2SLC6A3RENKCNH2
SCHEMBL662637 0.71 REN (0.47) SLC6A4SLC6A2SLC6A3RENKCNH2
SCHEMBL12837153 0.71 REN (0.80) RENKCNH2CYP3A4
SCHEMBL1518267 0.71 REN (0.80) RENKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009135299-A1 3, 4 - SUBSTITUTED PIPERIDINE DERIVATIVES AS RENIN INHIBITORS MERCK FROSST CANADA LTD. (CA) 2009-11-12 WO disclosed