SCHEMBL13625787

SCHEMBL13625787

CCCc1ccncc1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2E1 P05181 3/20 0.47
CYP2C8 P10632 3/20 0.47
CYP2D6 P10635 3/20 0.47
CYP2A6 P11509 3/20 0.47
CYP2C9 P11712 3/20 0.47
CYP2B6 P20813 3/20 0.47
CYP2C19 P33261 3/20 0.47
CYP3A4 P08684 3/20 0.43
CYP1A2 P05177 2/20 0.43
AOC1 P19801 4/20 0.41
AOC3 Q16853 4/20 0.41
PRKCI P41743 1/20 0.38
AURKA O14965 1/20 0.37
TYR P14679 2/20 0.37
HMGCR P04035 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
TDP1 Q9NUW8 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25774612 0.88 TYR (0.52) CYP2E1CYP2C8CYP2D6CYP2A6CYP2C9
SCHEMBL13625817 0.83
SCHEMBL5109069 0.82 CYP2E1 (0.46) CYP2E1CYP2C8CYP2D6CYP2A6CYP2C9
SCHEMBL10954433 0.80 CYP2E1 (0.51) CYP2E1CYP2C8CYP2D6CYP2A6CYP2C9
SCHEMBL28759090 0.79 TAAR1 (0.52) CYP2A6AOC1AOC3TDP1LOXL2
SCHEMBL6136671 0.78 PDE4B (0.40) AOC1AOC3TYRPDE4APDE4B
SCHEMBL5110078 0.78 CYP2E1 (0.46) CYP2E1CYP2C8CYP2D6CYP2A6CYP2C9
SCHEMBL7468680 0.77 CYP2E1 (0.49) CYP2E1CYP2C8CYP2D6CYP2A6CYP2C9
SCHEMBL8271491 0.77 CYP2E1 (0.49) CYP2E1CYP2C8CYP2D6CYP2A6CYP2C9
SCHEMBL873728 0.77 CYP2E1 (0.49) CYP2E1CYP2C8CYP2D6CYP2A6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009140448-A1 TETRAHYDROCYCLOPENTA[B]INDOLE ANDROGEN RECEPTOR MODULATORS ELI LILLY AND COMPANY (US) 2009-11-19 WO disclosed