SCHEMBL13625936

SCHEMBL13625936

NNc1cc2c3c(c1)C(c1ccccc1)CCN3CCC2c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
IDO1 P14902 1/20 0.34
CYP2C19 P33261 1/20 0.34
PTGS2 P35354 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
IGF1R P08069 1/20 0.34
ALOX15 P16050 1/20 0.34
DRD1 P21728 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2391384 0.83 DRD1 (0.43) IGF1RALOX15DRD1
SCHEMBL13625662 0.81 MAPT (0.43) LMNACYP3A4IDO1IGF1RALOX15
SCHEMBL8989689 0.79 SMN1; SMN2 (0.45) LMNA
SCHEMBL14523185 0.79 SCN9A (0.43) LMNA
SCHEMBL4347105 0.79 EEF2K (0.43)
SCHEMBL2391310 0.77 HTT (0.40) LMNA
SCHEMBL11997214 0.77 ALDH1A1 (0.35) IGF1RALOX15DRD1
SCHEMBL1411683 0.76 KDM4E (0.39) LMNA
SCHEMBL8988943 0.76 MAPT (0.39) LMNA
SCHEMBL13619991 0.76 NPC1 (0.48) LMNACYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009137342-A1 THERAPEUTICALLY USEFUL SUBSTITUTED 1, 7-DIPHENYL-L, 2, 3, 5, 6, 7-HEXAHYDROPYRIDO [ 3, 2, 1-I J ] QUINOLINE COMPOUNDS ALLERGAN, INC. (US) 2009-11-12 WO disclosed