SCHEMBL13626586

SCHEMBL13626586

CCN(c1cc(OC)ccc1C1CCc2cc(O)ccc2C1)C(C)c1ccc(OCCNC2CCCCC2)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.48
ESR2 Q92731 2/20 0.48
KDM4E B2RXH2 4/20 0.35
DRD2 P14416 4/20 0.32
DRD3 P35462 4/20 0.32
ALDH1A1 P00352 3/20 0.32
ADRA1D P25100 2/20 0.32
CYP26A1 O43174 1/20 0.31
DRD4 P21917 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
CNR2 P34972 1/20 0.31
XDH P47989 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13626585 0.92 ESR1 (0.49) ESR1ESR2DRD2DRD3ADRA1D
SCHEMBL13626576 0.91 ESR1 (0.52) ESR1ESR2KDM4EDRD2DRD3
SCHEMBL13626584 0.90 ESR1 (0.56) ESR1ESR2DRD2DRD3ADRA1D
SCHEMBL13626582 0.90 ESR1 (0.44) ESR1ESR2DRD2DRD3ADRA1D
SCHEMBL13626641 0.88 ESR1 (0.47) ESR1ESR2DRD2DRD3CYP26A1
SCHEMBL13626639 0.88 ESR1 (0.47) ESR1ESR2DRD2DRD3CYP26A1
SCHEMBL13626575 0.87 ESR1 (0.54) ESR1ESR2KDM4EDRD2DRD3
SCHEMBL13626660 0.86 ESR1 (0.45) ESR1ESR2DRD2DRD3CYP26A1
SCHEMBL13626640 0.86 ESR1 (0.46) ESR1ESR2DRD2DRD3CYP26A1
SCHEMBL13626642 0.85 ESR1 (0.45) ESR1ESR2DRD2DRD3CYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612114-B2 Such as (R)-6-{2-{ethyl[4-(2-ethylaminoethyl)benzyl]amino }-4-methoxyphenyl }-5,6,7,8-tetrahydronaphthalen-2-ol; osteoporosis; breast cancer EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-11-03 US disclosed