SCHEMBL13626708

SCHEMBL13626708

CCN(c1cc(OC)c(OC)cc1[C@@H]1CCc2cc(O)ccc2C1)C(C)c1ccc(OCCN2CCCCC2)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.38
ESR2 Q92731 5/20 0.36
HTR2C P28335 1/20 0.36
KDR P35968 2/20 0.36
CXCR3 P49682 4/20 0.35
CHEK1 O14757 2/20 0.35
MCHR1 Q99705 1/20 0.35
LTA4H P09960 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13626703 0.99 ESR1 (0.37) ESR1ESR2HTR2CKDRCXCR3
SCHEMBL13626711 0.94 HTR2C (0.36) ESR1ESR2HTR2CCXCR3
SCHEMBL13626675 0.90 ESR1 (0.44) ESR1ESR2HTR2C
SCHEMBL13626670 0.90 ESR1 (0.44) ESR1ESR2HTR2C
SCHEMBL13626668 0.89 ESR1 (0.43) ESR1ESR2HTR2C
SCHEMBL13626702 0.88 ESR1 (0.37) ESR1ESR2KDRCXCR3
SCHEMBL13626700 0.88 ESR1 (0.37) ESR1ESR2KDRCXCR3CHEK1
SCHEMBL13626638 0.86 ESR2 (0.44) ESR1ESR2HTR2C
SCHEMBL228649 0.85 ESR1 (0.48) ESR1ESR2HTR2CKDRCHEK1
SCHEMBL226461 0.85 ESR1 (0.48) ESR1ESR2HTR2CKDRCHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612114-B2 Such as (R)-6-{2-{ethyl[4-(2-ethylaminoethyl)benzyl]amino }-4-methoxyphenyl }-5,6,7,8-tetrahydronaphthalen-2-ol; osteoporosis; breast cancer EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-11-03 US disclosed