SCHEMBL13626711

SCHEMBL13626711

CCN(c1cc(OC)c(OC)cc1[C@@H]1CCc2cc(O)ccc2C1)C(C)c1ccc(OCCN2CCC(C)CC2)c(F)c1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 12/20 0.36
HTR2A P28223 8/20 0.36
HTR2B P41595 8/20 0.36
CXCR3 P49682 3/20 0.35
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
KDM4E B2RXH2 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13626703 0.94 ESR1 (0.37) HTR2CHTR2AHTR2BCXCR3ESR1
SCHEMBL13626708 0.94 ESR1 (0.38) HTR2CCXCR3ESR1ESR2
SCHEMBL13626638 0.93 ESR2 (0.44) HTR2CHTR2AHTR2BESR1ESR2
SCHEMBL13626673 0.90 ESR1 (0.42) HTR2CHTR2AHTR2BESR1ESR2
SCHEMBL13626702 0.87 ESR1 (0.37) CXCR3ESR1ESR2CYP2D6
SCHEMBL13626700 0.87 ESR1 (0.37) CXCR3ESR1ESR2CYP2D6
SCHEMBL228246 0.85 ESR1 (0.47) HTR2CHTR2AHTR2BCXCR3ESR1
SCHEMBL229625 0.85 ESR1 (0.47) HTR2CHTR2AHTR2BCXCR3ESR1
SCHEMBL13626668 0.84 ESR1 (0.43) HTR2CHTR2AHTR2BESR1ESR2
SCHEMBL13626670 0.83 ESR1 (0.44) HTR2CHTR2AHTR2BESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612114-B2 Such as (R)-6-{2-{ethyl[4-(2-ethylaminoethyl)benzyl]amino }-4-methoxyphenyl }-5,6,7,8-tetrahydronaphthalen-2-ol; osteoporosis; breast cancer EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-11-03 US disclosed