SCHEMBL13626995

SCHEMBL13626995

CC(C)(C)CC(=O)N1CCC(NC(=O)c2cccc3ccc(-c4cccc(C(F)(F)F)c4)nc23)CC1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 4/20 0.47
EPHX2 P34913 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
PHGDH O43175 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
JAK2 O60674 1/20 0.40
MAP4K4 O95819 2/20 0.40
GPR52 Q9Y2T5 1/20 0.39
KDM1A O60341 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
SYK P43405 1/20 0.39
MEN1 O00255 1/20 0.39
UBE2M P61081 1/20 0.39
KMT2A Q03164 1/20 0.39
DCUN1D1 Q96GG9 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17772313 0.92 DRD4 (0.46) DRD4EPHX2SMN1; SMN2ALDH1A1HPGD
SCHEMBL12880950 0.87 PARP1 (0.50) DRD4SMN1; SMN2ALDH1A1HPGDMAPT
SCHEMBL1035236 0.84 MAPT (0.50) DRD4EPHX2SMN1; SMN2ALDH1A1MAPT
SCHEMBL1034071 0.81 CNR2 (0.49) DRD4MAPTMAP4K4GPR52KDM1A
SCHEMBL1032826 0.81 POLB (0.45) DRD4MAPTJAK2MAP4K4KDM1A
SCHEMBL1033395 0.78 HDAC4 (0.46) DRD4MAP4K4MEN1KMT2A
SCHEMBL1033396 0.78 HDAC4 (0.46) DRD4MAP4K4MEN1KMT2A
SCHEMBL1032402 0.77 CHRNA7 (0.52)
SCHEMBL1034785 0.74 SCN7A (0.42) DRD4MAP4K4GPR52KDM1A
SCHEMBL4602598 0.73 EPHX2 (0.60) DRD4EPHX2PHGDHMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134973-A1 QUENOLINES AND RELATED ANALOGS AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed