SCHEMBL13627346

SCHEMBL13627346

c1ccc2c(c1)NC[C@H]1CNC[C@@H]21

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 2/20 0.41
CHRNA3 P32297 2/20 0.41
HTR2C P28335 6/20 0.38
HTR2A P28223 3/20 0.38
HTR2B P41595 3/20 0.38
BPTF Q12830 1/20 0.36
CHRNB2 P17787 3/20 0.33
CHRNA4 P43681 3/20 0.33
CHRNA7 P36544 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4399620 1.00 CHRNB4 (0.41) CHRNB4CHRNA3HTR2CHTR2AHTR2B
SCHEMBL14411860 0.94 CHRNB4 (0.42) CHRNB4CHRNA3HTR2CHTR2AHTR2B
SCHEMBL1804494 0.84 CHRNB4 (0.37) CHRNB4CHRNA3HTR2CHTR2AHTR2B
SCHEMBL1804493 0.84 CHRNB4 (0.37) CHRNB4CHRNA3HTR2CHTR2AHTR2B
SCHEMBL1804490 0.84 CHRNB4 (0.37) CHRNB4CHRNA3HTR2CHTR2AHTR2B
SCHEMBL24138192 0.80 CHRNB4 (0.39) CHRNB4CHRNA3HTR2CHTR2BCHRNB2
SCHEMBL19696035 0.80 CHRNB4 (0.39) CHRNB4CHRNA3HTR2CHTR2BCHRNB2
SCHEMBL19122664 0.80 CHRNB4 (0.39) CHRNB4CHRNA3HTR2CHTR2BCHRNB2
SCHEMBL30417082 0.79 CHRNB4 (0.39) CHRNB4CHRNA3
SCHEMBL18925342 0.78 MEN1 (0.35) CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7618980-B2 Pyrrolo(oxo)quinolines as 5HT ligands BRISTOL-MYERS SQUIBB COMPANY (US) 2009-11-17 US disclosed
US-7618980-B2 Pyrrolo(oxo)quinolines as 5HT ligands BRISTOL-MYERS SQUIBB COMPANY (US) 2009-11-17 US disclosed