SCHEMBL13628749

SCHEMBL13628749

Cc1ncc(-c2cnn[nH]2)o1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.37
CA2 P00918 5/20 0.37
CA9 Q16790 5/20 0.37
CA1 P00915 4/20 0.37
LRRK2 Q5S007 1/20 0.33
PIK3CG P48736 1/20 0.32
HDAC4 P56524 1/20 0.31
ADRA1A P35348 1/20 0.30
PDK2 Q15119 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13628728 0.77 NOTUM (0.31)
SCHEMBL13628747 0.73 MAPT (0.41)
SCHEMBL13628742 0.65 CA12 (0.37) CA12CA2CA9CA1LRRK2
SCHEMBL13484011 0.63 CA12 (0.41) CA12CA2CA9CA1LRRK2
SCHEMBL13628752 0.61 NPSR1 (0.34)
SCHEMBL5020173 0.61 CCR1 (0.56)
SCHEMBL9284900 0.61 CA12 (0.61) CA12CA2CA9CA1LRRK2
SCHEMBL5020207 0.61 NPC1 (0.59) CA2CA9CA1
SCHEMBL17791784 0.60
SCHEMBL13411815 0.60 POLB (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed
US-7612070-B2 Heterocyclic compounds as antiinflammatory agents and cyclooxygenase inhibitors CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2009-11-03 US disclosed