SCHEMBL13630537

SCHEMBL13630537

C=C(COc1ccccc1-c1cc(C(N)=O)c(NC(N)=O)[nH]1)OC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 5/20 0.45
CHUK O15111 2/20 0.41
INSR P06213 2/20 0.41
MAPK8 P45983 2/20 0.41
CAMKK2 Q96RR4 2/20 0.41
MAPT P10636 4/20 0.40
RAB9A P51151 4/20 0.40
NPC1 O15118 3/20 0.40
TP53 P04637 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CDC7 O00311 1/20 0.40
IKBKB O14920 1/20 0.38
CASP3 P42574 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
ALDH1A1 P00352 2/20 0.36
PARP1 P09874 1/20 0.35
NR3C2 P08235 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2199592 0.89 BRD4 (0.46) BRD4CHUKINSRMAPK8CAMKK2
SCHEMBL2197555 0.85 BRD4 (0.49) BRD4CHUKINSRMAPK8CAMKK2
SCHEMBL2200493 0.84 BRD4 (0.46) BRD4CHUKINSRMAPK8CAMKK2
SCHEMBL2196927 0.84 CDC7 (0.54) BRD4CHUKINSRMAPK8CAMKK2
SCHEMBL2198470 0.83 BRD4 (0.47) BRD4CHUKINSRMAPK8CAMKK2
SCHEMBL12509787 0.82 KMT2A (0.50) BRD4CHUKINSRMAPK8CAMKK2
SCHEMBL2199883 0.82 CHEK1 (0.45) BRD4CHUKINSRMAPK8CAMKK2
SCHEMBL2195870 0.81 KDM4E (0.50) BRD4CHUKINSRMAPK8CAMKK2
SCHEMBL2199427 0.81 MAPT (0.55) BRD4CHUKINSRMAPK8CAMKK2
SCHEMBL2197053 0.81 BRD4 (0.47) BRD4IKBKBPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2116530-A1 NOVEL PYRROLE DERIVATIVE HAVING UREIDE GROUP AND AMINOCARBONYL GROUP AS SUBSTITUENTS Santen Pharmaceutical Co., Ltd (JP) 2009-11-11 EP disclosed