SCHEMBL13634118

SCHEMBL13634118

CN(C)Cc1nc(Br)c(C(=O)NCc2ccc(Cl)c(Oc3cc(Cl)cc(C#N)c3)c2F)[nH]1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.45
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KCNH2 Q12809 2/20 0.34
PTGES O14684 11/20 0.32
EPHX2 P34913 1/20 0.32
MEP1B Q16820 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL13560338 0.96 CYP3A4 (0.42) CYP3A4CYP2C9CYP2C19KCNH2PTGES
SCHEMBL3033183 0.92 CYP3A4 (0.46) CYP3A4CYP2C9CYP2C19KCNH2PTGES
SCHEMBL3800799 0.92 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19KCNH2PTGES
SCHEMBL3639074 0.91 CYP3A4 (0.46) CYP3A4CYP2C9CYP2C19KCNH2PTGES
SCHEMBL13638743 0.91 CYP3A4 (0.43) CYP3A4CYP2C9CYP2C19KCNH2EPHX2
SCHEMBL3638768 0.90 CYP3A4 (0.46) CYP3A4CYP2C9CYP2C19KCNH2PTGES
SCHEMBL3805676 0.90 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19KCNH2PTGES
SCHEMBL3639944 0.89 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19KCNH2PTGES
SCHEMBL3031620 0.89 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19KCNH2PTGES
SCHEMBL13982119 0.89 PTGES (0.35) PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8304419-B2 Chemical compounds GLAXOSMITHKLINE LLC (US) 2012-11-06 US disclosed
US-8304419-B2 Chemical compounds GLAXOSMITHKLINE LLC (US) 2012-11-06 US disclosed