SCHEMBL13634923

SCHEMBL13634923

CCCNC(=O)c1cc(CN2CCNC[C@@H]2C)ccc1NC(=O)c1csc(N2CC[C@H](OC)C2)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 14/20 0.36
GLS O94925 1/20 0.36
HDAC3 O15379 1/20 0.34
HDAC2 Q92769 1/20 0.34
SCD O00767 2/20 0.34
SCD5 Q86SK9 2/20 0.34
PARP1 P09874 1/20 0.34
TNK1 Q13470 1/20 0.34
MAPKAPK2 P49137 1/20 0.33
JAK2 O60674 1/20 0.33
ROCK2 O75116 1/20 0.33
IGF1R P08069 1/20 0.33
MAPK1 P28482 1/20 0.33
AKT1 P31749 1/20 0.33
RPS6KA3 P51812 1/20 0.33
NEK2 P51955 1/20 0.33
STK3 Q13188 1/20 0.33
CAMK4 Q16566 1/20 0.33
TSSK2 Q96PF2 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13634574 1.00 CHEK1 (0.36) CHEK1GLSHDAC3HDAC2SCD
SCHEMBL13164118 0.95 CHEK1 (0.36) CHEK1HDAC3HDAC2SCDSCD5
SCHEMBL13270439 0.95 CHEK1 (0.36) CHEK1HDAC3HDAC2SCDSCD5
SCHEMBL13634732 0.93 CHEK1 (0.35) CHEK1HDAC3HDAC2SCDSCD5
SCHEMBL13634669 0.89 GLS (0.35) CHEK1GLSSCDSCD5PARP1
SCHEMBL13634768 0.89 GLS (0.35) CHEK1GLSSCDSCD5PARP1
SCHEMBL13634906 0.88 SCD (0.38) CHEK1GLSSCDSCD5PARP1
SCHEMBL13634750 0.88 IRAK4 (0.38) GLSSCDSCD5IRAK4
SCHEMBL13634760 0.86 GLS (0.40) CHEK1GLSSCDSCD5
SCHEMBL13634751 0.86 GLS (0.39) CHEK1GLSSCDSCD5PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8304547-B2 Azolecarboxamide compound or salt thereof ASTELLAS PHARMA INC. (JP) 2012-11-06 US disclosed