SCHEMBL13635206

SCHEMBL13635206

C=Cc1ccc(-n2c(C)cc(CCCc3ccc(F)cc3F)cc2=O)c(C)c1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 16/20 0.36
GSK3B P49841 1/20 0.33
BACE1 P56817 1/20 0.33
DAO P14920 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ROCK2 O75116 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
STRADA Q7RTN6 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4376213 0.80 MAPK14 (0.45) MAPK14GSK3BBACE1ROCK2MAPK12
SCHEMBL13635776 0.79 MAPK14 (0.48) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL6471335 0.73 MAPK14 (0.47) MAPK14GSK3BBACE1ROCK2MAPK12
SCHEMBL29594177 0.72 MAPK14 (0.68) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL4376529 0.72 MAPK14 (0.68) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL3526705 0.67 MAPK14 (0.48) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL4468565 0.64 MAPK14 (0.50) MAPK14GSK3BBACE1
SCHEMBL4376549 0.64 MAPK14 (0.52) MAPK14ROCK2MAPK12MAPK11STRADA
SCHEMBL27699486 0.63 TYR (0.43)
SCHEMBL13610118 0.62 GSK3B (0.47) MAPK14GSK3BBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490064-B1 SUBSTITUTED PYRIDINONES AS MODULATORS OF P38 MAP KINASE PHARMACIA CORP (US) 2009-11-18 EP disclosed