SCHEMBL13635258

SCHEMBL13635258

CS(=O)(=O)c1ccc(/C(COC(=O)OCC(CON(O)O)ON(O)O)=C(/C(=O)OCc2ccccc2)c2ccccc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.35
MAPT P10636 1/20 0.34
ESR2 Q92731 3/20 0.33
PTPN1 P18031 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13635052 0.91 PTGS2 (0.38) PTGS2ESR2
SCHEMBL14045665 0.90 PTGS2 (0.37) PTGS2MAPTESR2PTPN1
SCHEMBL13635220 0.89 PTGS2 (0.38) PTGS2ESR2
SCHEMBL13635600 0.83 PTGS2 (0.35) PTGS2ESR2
SCHEMBL13635257 0.82 ESR2 (0.35) PTGS2ESR2
SCHEMBL13624620 0.81 PTGS2 (0.43) PTGS2MAPTESR2
SCHEMBL14025307 0.81 ESR2 (0.42) PTGS2MAPTESR2
SCHEMBL14045664 0.81 PTGS2 (0.41) PTGS2ESR2
SCHEMBL13635256 0.80 ESR2 (0.36) PTGS2ESR2
SCHEMBL13632531 0.80 PTGS2 (0.38) PTGS2ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622501-B2 Nitric oxide releasing prodrugs of diaryl-2-(5H)-furanones as cyclooxygenase-2 inhibitors MERCK FROSST CANADA & CO. (CA) 2009-11-24 US disclosed