SCHEMBL13635913

SCHEMBL13635913

Bc1c(O)cc(C)n(-c2cc(C(=O)NC)ccc2C(=O)OC)c1=O

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
LMNA P02545 1/20 0.50
MYC P01106 8/20 0.41
MAPK14 Q16539 7/20 0.39
ROCK2 O75116 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
STRADA Q7RTN6 1/20 0.38
TSHR P16473 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA7 P43166 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK4 Q16654 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4390396 0.87 ALDH1A1 (0.50) ALDH1A1LMNAMYCMAPK14ROCK2
SCHEMBL4379220 0.81 ALDH1A1 (0.50) ALDH1A1LMNAMYCMAPK14ROCK2
SCHEMBL6646966 0.75 MYC (0.51) MYCMAPK14ROCK2MAPK12MAPK11
SCHEMBL14189583 0.71 ALDH1A1 (0.53) ALDH1A1MYC
SCHEMBL2706592 0.71 MAPK14 (0.57) ALDH1A1MAPK14ROCK2MAPK12MAPK11
SCHEMBL12268010 0.70 KDM4E (0.50) ALDH1A1MAPK14TSHRCA12CA1
SCHEMBL15668584 0.70 MYC (0.75) ALDH1A1LMNAMYC
SCHEMBL15714708 0.69 MYC (0.60) ALDH1A1LMNAMYC
Hydrazine SCHEMBL15668725 0.69 MYC (0.73) ALDH1A1LMNAMYC
SCHEMBL4377764 0.68 ALDH1A1 (0.52) ALDH1A1LMNAMYCTSHRCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1490064-B1 SUBSTITUTED PYRIDINONES AS MODULATORS OF P38 MAP KINASE PHARMACIA CORP (US) 2009-11-18 EP disclosed