SCHEMBL13636798

SCHEMBL13636798

Bc1ccc(C(=O)NCCC)s1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.50
POLB P06746 4/20 0.50
RAB9A P51151 4/20 0.50
NPC1 O15118 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
GAA P10253 2/20 0.50
ESR1 P03372 2/20 0.50
MAPT P10636 2/20 0.50
HPGD P15428 2/20 0.50
JMJD7 P0C870 1/20 0.50
STAT3 P40763 1/20 0.50
STAT1 P42224 1/20 0.50
RXFP1 Q9HBX9 2/20 0.47
NPSR1 Q6W5P4 1/20 0.47
MAPK1 P28482 1/20 0.45
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
ALDH1A1 P00352 3/20 0.44
GFER P55789 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27547515 0.82 GAA (0.54) KDM4EPOLBRAB9ANPC1SMN1; SMN2
SCHEMBL6360616 0.81 GSK3B (0.53) KDM4EPOLBRAB9ANPC1SMN1; SMN2
SCHEMBL1587164 0.81 KDM4E (0.51) KDM4EPOLBRAB9ANPC1SMN1; SMN2
SCHEMBL12124267 0.81 POLB (0.65) KDM4EPOLBRAB9ANPC1SMN1; SMN2
SCHEMBL6362085 0.79 GAA (0.75) KDM4EPOLBRAB9ANPC1SMN1; SMN2
SCHEMBL12313385 0.79 RAB9A (0.60) KDM4EPOLBRAB9ANPC1SMN1; SMN2
SCHEMBL6977403 0.79 KDM4E (0.50) KDM4EPOLBRAB9ANPC1SMN1; SMN2
SCHEMBL6362178 0.79 MAPK1 (0.69) KDM4EPOLBRAB9ANPC1SMN1; SMN2
SCHEMBL2001834 0.78 NPSR1 (0.50) KDM4EPOLBRAB9ANPC1SMN1; SMN2
SCHEMBL6978678 0.78 KDM4E (0.49) KDM4EPOLBRAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009137081-A2 SMALL MOLECULE INHIBITORS OF PLASMODIUM FALCIPARUM DIHYDROOROTATE DEHYDROGENASE MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2009-11-12 WO disclosed