SCHEMBL13636993

SCHEMBL13636993

CCCNC(=O)c1ccc(-n2ccc3c2C=CCC3)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.43
ACKR3 P25106 5/20 0.40
KDM4E B2RXH2 4/20 0.39
MAPT P10636 3/20 0.39
HPGD P15428 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GFER P55789 1/20 0.39
POLB P06746 3/20 0.36
GAA P10253 2/20 0.36
ESR1 P03372 2/20 0.36
NPC1 O15118 1/20 0.36
JMJD7 P0C870 1/20 0.36
STAT3 P40763 1/20 0.36
STAT1 P42224 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
RXFP1 Q9HBX9 3/20 0.34
DHODH Q02127 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
SHMT2 P34897 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13636799 0.83 MAPT (0.42) HTR2CACKR3KDM4EMAPTHPGD
SCHEMBL13636931 0.82 ACKR3 (0.39) HTR2CACKR3KDM4EMAPTHPGD
SCHEMBL1948468 0.71 HTR2C (0.77) HTR2CACKR3KDM4EMAPTHPGD
SCHEMBL1946018 0.70 HDAC8 (0.46) ACKR3KDM4EMAPTHPGDALDH1A1
SCHEMBL1945680 0.70 RXFP1 (0.55) HTR2CACKR3KDM4EMAPTHPGD
SCHEMBL1945681 0.69 RXFP1 (0.57) HTR2CACKR3KDM4EMAPTHPGD
SCHEMBL1949315 0.68 ACKR3 (0.76) HTR2CACKR3KDM4EMAPTHPGD
SCHEMBL1946478 0.67 MEN1 (0.50) ACKR3KDM4EMAPTHPGDALDH1A1
SCHEMBL1944624 0.66 NAMPT (0.51) HTR2CACKR3KDM4EMAPTHPGD
SCHEMBL1948464 0.66 KDM4E (0.46) HTR2CACKR3KDM4EMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009137081-A2 SMALL MOLECULE INHIBITORS OF PLASMODIUM FALCIPARUM DIHYDROOROTATE DEHYDROGENASE MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2009-11-12 WO disclosed