SCHEMBL13637689

SCHEMBL13637689

C[C@H]1CCC(=O)N2CCC[C@@H](C(=O)N[C@@H](CC(=O)O)C(=O)c3ncc(-c4c(Cl)cccc4Cl)o3)N2C1=O

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 8/20 0.42
CASP3 P42574 4/20 0.42
IL1B P01584 2/20 0.40
MME P08473 1/20 0.34
ACE P12821 1/20 0.34
LCK P06239 7/20 0.34
GZMB P10144 1/20 0.33
CASP8 Q14790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL647407 0.89 CASP1 (0.44) CASP1CASP3IL1BMMEACE
SCHEMBL645919 0.89 CASP1 (0.44) CASP1CASP3IL1BMMEACE
SCHEMBL10200732 0.85 CASP1 (0.47) CASP1CASP3IL1BMMEACE
SCHEMBL10199394 0.84 CASP1 (0.43) CASP1CASP3IL1BGZMBCASP8
SCHEMBL10251411 0.84 CASP1 (0.43) CASP1CASP3IL1BGZMBCASP8
SCHEMBL7735511 0.81 CASP1 (0.37) CASP1CASP3IL1BLCKCASP8
SCHEMBL646048 0.75 CASP1 (0.45) CASP1CASP3IL1BMMEACE
SCHEMBL645261 0.71 CASP1 (0.59) CASP1CASP3IL1BMMEACE
SCHEMBL648084 0.71 CASP1 (0.59) CASP1CASP3IL1BMMEACE
SCHEMBL644683 0.70 CASP1 (0.41) CASP1CASP3IL1BMMEACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2123665-A2 Inhibitors of interleukin-1Beta converting enzyme Vertex Pharmaceuticals Incorporated (US) 2009-11-25 EP disclosed