SCHEMBL13637705

SCHEMBL13637705

C=C/C(Cl)=C(\C=C/C)CSCC(=O)[C@H](CC(=O)O)NC(=O)Cn1c(Cc2ccccc2)ccc(NC(=O)CCc2ccccc2)c1=O

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 16/20 0.57
IL1B P01584 4/20 0.57
ELANE P08246 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12450466 0.80 CASP1 (0.61) CASP1IL1B
SCHEMBL12450458 0.80 CASP1 (0.71) CASP1IL1BELANE
SCHEMBL951210 0.79 CASP1 (0.73) CASP1IL1BELANE
SCHEMBL645752 0.73 CASP1 (0.62) CASP1IL1B
SCHEMBL12914456 0.73 CASP1 (0.62) CASP1IL1B
SCHEMBL4459947 0.73 CASP1 (1.00) CASP1IL1BELANE
SCHEMBL12450638 0.73 CASP1 (1.00) CASP1IL1BELANE
SCHEMBL950212 0.73 CASP1 (0.61) CASP1IL1BELANE
SCHEMBL12450470 0.73 CASP1 (0.61) CASP1IL1BELANE
SCHEMBL949357 0.71 CASP1 (0.60) CASP1IL1BELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2123665-A2 Inhibitors of interleukin-1Beta converting enzyme Vertex Pharmaceuticals Incorporated (US) 2009-11-25 EP disclosed