SCHEMBL13637751

SCHEMBL13637751

O=C[C@H](CC(=O)O)NC(=O)CN1C(=O)[C@@H](NC(=O)CCc2ccccc2)CN(C(=O)CCc2ccccc2)c2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 10/20 0.53
IL1B P01584 4/20 0.47
XIAP P98170 5/20 0.47
CYP3A4 P08684 4/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12914484 0.93 CASP1 (0.52) CASP1IL1BXIAPCYP3A4
SCHEMBL646010 0.93 CASP1 (0.63) CASP1IL1BXIAPCYP3A4
SCHEMBL646012 0.93 CASP1 (0.63) CASP1IL1BXIAPCYP3A4
SCHEMBL10247704 0.91 CASP1 (0.49) CASP1IL1BXIAPCYP3A4
SCHEMBL10199246 0.91 CASP1 (0.49) CASP1IL1BXIAPCYP3A4
SCHEMBL650470 0.89 CASP1 (0.50) CASP1IL1BXIAPCYP3A4
SCHEMBL647991 0.88 CASP1 (0.50) CASP1IL1BXIAPCYP3A4
SCHEMBL647990 0.88 CASP1 (0.50) CASP1IL1BXIAPCYP3A4
SCHEMBL647989 0.88 CASP1 (0.50) CASP1IL1BXIAPCYP3A4
SCHEMBL10249689 0.86 CASP1 (0.61) CASP1XIAPCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2123665-A2 Inhibitors of interleukin-1Beta converting enzyme Vertex Pharmaceuticals Incorporated (US) 2009-11-25 EP disclosed