SCHEMBL13637760

SCHEMBL13637760

O=C[C@H](CC(=O)O)NC(=O)CN1CCN(Cc2ccccc2)C[C@H](NC(=O)OCc2ccccc2)C1=O

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 8/20 0.55
CASP3 P42574 3/20 0.44
CASP9 P55211 2/20 0.42
CASP8 Q14790 2/20 0.42
F2 P00734 5/20 0.41
F10 P00742 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL948554 0.95 CASP1 (0.51) CASP1CASP3CASP9CASP8F2
Trifluoroacetic Acid SCHEMBL948555 0.95 CASP1 (0.51) CASP1CASP3CASP9CASP8F2
SCHEMBL12450523 0.94 CASP1 (0.47) CASP1CASP3CASP9CASP8F2
SCHEMBL12450947 0.87 CASP1 (0.55) CASP1CASP3CASP9CASP8F2
SCHEMBL14370034 0.84 CASP1 (0.53) CASP1CASP3CTSLCTSB
SCHEMBL13547350 0.82 SMN1; SMN2 (0.47) CASP3CTSLCTSB
SCHEMBL949976 0.81 CASP1 (0.53) CASP1CTSLCTSB
SCHEMBL12914629 0.81 CASP1 (0.53) CASP1CTSLCTSB
SCHEMBL14370035 0.81 CASP1 (0.53) CASP1CTSLCTSB
Trifluoroacetic Acid SCHEMBL948894 0.80 CASP1 (0.49) CASP1CTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2123665-A2 Inhibitors of interleukin-1Beta converting enzyme Vertex Pharmaceuticals Incorporated (US) 2009-11-25 EP disclosed