SCHEMBL13638417

SCHEMBL13638417

C=C1CC(Nc2ncc(C)c(-c3ccc(CCCCO)s3)n2)CC(C)(C)N1

nearest known ligand 0.31

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.31
CHUK O15111 1/20 0.31
IKBKG Q9Y6K9 1/20 0.31
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4494160 0.89 IKBKB (0.33) IKBKBCHUKIKBKGMAPK1
SCHEMBL13638661 0.88 RPS6KB2 (0.38)
SCHEMBL13638303 0.86 IKBKB (0.43) IKBKBCHUKIKBKG
SCHEMBL13638505 0.81 JUN (0.31) MAPK1
SCHEMBL3471753 0.79 IKBKB (0.32) IKBKBCHUKIKBKG
SCHEMBL13638415 0.77 CDK7 (0.34) IKBKBCHUKIKBKG
SCHEMBL4482123 0.77 RPS6KB2 (0.41) MAPK1
SCHEMBL13638292 0.76 KDR (0.37) IKBKBCHUKIKBKG
SCHEMBL13638316 0.76 KCNH2 (0.44) MAPK1
SCHEMBL13638306 0.76 IKBKB (0.34) IKBKBCHUKIKBKG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7615562-B2 Such as 2-methyl-4-{5-[2-(2,2,6,6-tetramethyl-piperidin-4-ylamino)-pyrimidin-4-yl]-thiophen-2-yl}-butan-2-ol; tumor necrosis factor inhibitors; immunosuppressants; antiinflammatory agents NOVARTIS AG (CH) 2009-11-10 US disclosed