SCHEMBL13638466

SCHEMBL13638466

C=C1CC(Nc2nccc(-c3ccc(C(=O)NCCc4ccccc4)s3)n2)CC(C)(C)N1

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKT3 Q9Y243 13/20 0.62
HDAC1 Q13547 4/20 0.40
GAA P10253 1/20 0.39
TEC P42680 1/20 0.39
TXK P42681 1/20 0.39
BTK Q06187 1/20 0.39
ITK Q08881 1/20 0.39
NPC1 O15118 1/20 0.38
USP2 O75604 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13638474 0.92 AKT3 (0.50) AKT3HDAC1TECTXKBTK
SCHEMBL3477527 0.89 AKT3 (0.68) AKT3HDAC1GAARAB9A
SCHEMBL13638295 0.85 AKT3 (0.38) AKT3GAATECTXKBTK
SCHEMBL13638465 0.85 HPGDS (0.47) AKT3TECTXKBTKITK
SCHEMBL13638504 0.84 AKT3 (0.48) AKT3GAATECTXKBTK
SCHEMBL13638565 0.84 AKT3 (0.48) AKT3GAATECTXKBTK
SCHEMBL14612850 0.82 AKT3 (0.37) AKT3TECTXKBTKITK
SCHEMBL13638430 0.81 AKT3 (0.36) AKT3
SCHEMBL13638669 0.81 CDK2 (0.36) AKT3TECTXKBTKITK
SCHEMBL13638569 0.80 AKT3 (0.37) AKT3TECTXKBTKITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7615562-B2 Such as 2-methyl-4-{5-[2-(2,2,6,6-tetramethyl-piperidin-4-ylamino)-pyrimidin-4-yl]-thiophen-2-yl}-butan-2-ol; tumor necrosis factor inhibitors; immunosuppressants; antiinflammatory agents NOVARTIS AG (CH) 2009-11-10 US disclosed