SCHEMBL13638528

SCHEMBL13638528

Nc1ccc2c(=O)n(-c3c(F)cc(C(=O)NS(=O)(=O)c4ccc(Cl)s4)cc3CF)c(=O)[nH]c2c1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 2/20 0.46
TP53 P04637 1/20 0.35
HTR3A P46098 2/20 0.32
RXFP1 Q9HBX9 1/20 0.32
PPARG P37231 1/20 0.31
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13638527 0.88 P2RY12 (0.45) P2RY12TP53HTR3ARXFP1AKR1C3
SCHEMBL6017209 0.82 P2RY12 (0.54) P2RY12TP53HTR3ARXFP1MAPT
SCHEMBL9922414 0.82 P2RY12 (0.58) P2RY12TP53HTR3ARXFP1MAPT
SCHEMBL12161684 0.80 P2RY12 (0.56) P2RY12TP53MAPT
SCHEMBL17715382 0.80 P2RY12 (0.49) P2RY12TP53HTR3ARXFP1PPARG
SCHEMBL13638520 0.79 P2RY12 (0.47) P2RY12TP53RXFP1MAPT
SCHEMBL13638523 0.79 P2RY12 (0.55) P2RY12TP53HTR3ARXFP1MAPT
SCHEMBL9923005 0.77 P2RY12 (0.54) P2RY12TP53PPARGMAPT
SCHEMBL9922413 0.74 P2RY12 (0.59) P2RY12TP53HTR3ARXFP1MAPT
SCHEMBL4412669 0.74 P2RY12 (0.70) P2RY12TP53RXFP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622474-B2 Asulfonyl(urea, thiourea, guanidine, cyanoguanidine) compounds; cardiovascular disorders; thrombosis PORTOLA PHARMACEUTICALS, INC. (US) 2009-11-24 US disclosed