SCHEMBL13638533

SCHEMBL13638533

C=C1CC(Nc2nccc(-c3ccc(Br)cc3)n2)CC(C)(C)N1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 11/20 0.43
PIK3CG P48736 6/20 0.40
PIK3CA P42336 5/20 0.40
PIK3CB P42338 5/20 0.40
MAPK8 P45983 2/20 0.39
HDAC8 Q9BY41 1/20 0.38
CDK1 P06493 1/20 0.37
CDK4 P11802 1/20 0.37
CCNB1 P14635 1/20 0.37
CCNA2 P20248 1/20 0.37
CCND1 P24385 1/20 0.37
CDK2 P24941 1/20 0.37
CCNA1 P78396 1/20 0.37
MAPK9 P45984 1/20 0.37
MAPK10 P53779 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14612807 0.90 IKBKB (0.44) IKBKBMAPK8HDAC8CDK1CDK4
SCHEMBL13638440 0.89 IKBKB (0.43) IKBKBMAPK8HDAC8CDK1CDK4
SCHEMBL13638678 0.89 IKBKB (0.42) IKBKBMAPK8HDAC8CDK1CDK4
SCHEMBL14612854 0.87 IKBKB (0.42) IKBKBMAPK8HDAC8CDK1CDK4
SCHEMBL13638436 0.87 IKBKB (0.42) IKBKBMAPK8HDAC8CDK1CDK4
SCHEMBL14612808 0.86 HDAC8 (0.44) IKBKBMAPK8HDAC8
SCHEMBL13638679 0.85 IKBKB (0.41) IKBKBMAPK8CDK1CDK4CCNB1
SCHEMBL13638478 0.85 IKBKB (0.48) IKBKBMAPK8CDK4CDK2MAPK9
SCHEMBL13638584 0.84 KCNH2 (0.47) IKBKBHDAC8MAPK10
SCHEMBL3470852 0.84 IKBKB (0.48) IKBKBPIK3CGPIK3CAPIK3CBMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7615562-B2 Such as 2-methyl-4-{5-[2-(2,2,6,6-tetramethyl-piperidin-4-ylamino)-pyrimidin-4-yl]-thiophen-2-yl}-butan-2-ol; tumor necrosis factor inhibitors; immunosuppressants; antiinflammatory agents NOVARTIS AG (CH) 2009-11-10 US disclosed
US-20070043048-A1 2-Aminopyrimidine derivatives and their medical use NOVARTIS AG (CH) 2007-02-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070043048-A1 2-Aminopyrimidine derivatives and their medical use TPMT, IKBKB, CHUK IKBKB 2/4885PIK3CG 266/4885PIK3CA 132/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.