SCHEMBL13638478

SCHEMBL13638478

C=C1CC(Nc2nccc(-c3ccc(S(N)(=O)=O)cc3)n2)CC(C)(C)N1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 17/20 0.48
MAPK8 P45983 3/20 0.47
MAPK10 P53779 2/20 0.46
CHUK O15111 2/20 0.46
MAPK9 P45984 1/20 0.46
MAPK11 Q15759 1/20 0.46
MAPK14 Q16539 1/20 0.46
CDK4 P11802 1/20 0.43
CDK2 P24941 1/20 0.43
JAK2 O60674 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14612876 0.91 IKBKB (0.45) IKBKBMAPK8MAPK10CHUKMAPK9
SCHEMBL14612807 0.86 IKBKB (0.44) IKBKBMAPK8MAPK10MAPK9CDK4
SCHEMBL3471961 0.86 MEN1 (0.53) IKBKBMAPK8MAPK10CHUKMAPK9
SCHEMBL13638533 0.85 IKBKB (0.43) IKBKBMAPK8MAPK10MAPK9CDK4
SCHEMBL13638440 0.85 IKBKB (0.43) IKBKBMAPK8MAPK10MAPK9CDK4
SCHEMBL13638678 0.84 IKBKB (0.42) IKBKBMAPK8MAPK14CDK4CDK2
SCHEMBL14612854 0.83 IKBKB (0.42) IKBKBMAPK8MAPK10MAPK9CDK4
SCHEMBL13638436 0.83 IKBKB (0.42) IKBKBMAPK8MAPK10CHUKMAPK9
SCHEMBL13638562 0.83 IKBKB (0.39) IKBKBMAPK8MAPK10CHUKMAPK9
SCHEMBL13638679 0.82 IKBKB (0.41) IKBKBMAPK8MAPK10CHUKMAPK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7615562-B2 Such as 2-methyl-4-{5-[2-(2,2,6,6-tetramethyl-piperidin-4-ylamino)-pyrimidin-4-yl]-thiophen-2-yl}-butan-2-ol; tumor necrosis factor inhibitors; immunosuppressants; antiinflammatory agents NOVARTIS AG (CH) 2009-11-10 US disclosed