SCHEMBL13638928

SCHEMBL13638928

COCCN(C)c1nc(C(=O)Nc2ccc(CN3CCC[C@@H]3COC)cc2C(=O)OOC)cs1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.48
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC1 Q13547 1/20 0.44
DRD2 P14416 2/20 0.35
VEGFA P15692 1/20 0.34
EGLN1 Q9GZT9 1/20 0.34
MBTPS1 Q14703 1/20 0.34
AURKA O14965 1/20 0.33
RPS6KB1 P23443 1/20 0.33
MAP4K1 Q92918 1/20 0.33
SPHK2 Q9NRA0 1/20 0.33
SPHK1 Q9NYA1 1/20 0.33
ENPP2 Q13822 3/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13634788 0.95 S1PR1 (0.48) S1PR1HDAC8HDAC6HDAC1DRD2
SCHEMBL13634780 0.92 S1PR1 (0.48) S1PR1HDAC8HDAC6HDAC1VEGFA
SCHEMBL13634595 0.90 S1PR1 (0.49) S1PR1HDAC8HDAC6HDAC1DRD2
SCHEMBL13638884 0.90 S1PR1 (0.47) S1PR1HDAC8HDAC6HDAC1DRD2
SCHEMBL13270723 0.84 S1PR1 (0.42) S1PR1HDAC8HDAC6HDAC1VEGFA
SCHEMBL13162957 0.83 S1PR1 (0.42) S1PR1HDAC8HDAC6HDAC1DRD2
SCHEMBL13270438 0.81 ADORA2A (0.38) S1PR1MAP4K1
SCHEMBL13638887 0.80 S1PR1 (0.47) S1PR1HDAC8HDAC6HDAC1DRD2
SCHEMBL13638782 0.80 JAK2 (0.36) S1PR1
SCHEMBL13634841 0.80 S1PR1 (0.49) S1PR1HDAC8HDAC6HDAC1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8304547-B2 Azolecarboxamide compound or salt thereof ASTELLAS PHARMA INC. (JP) 2012-11-06 US disclosed