SCHEMBL13634841

SCHEMBL13634841

CCCNC(=O)c1cc(CN2CCC[C@@H]2COC)ccc1NC(=O)c1csc(N(C)CC2CCOCC2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 4/20 0.49
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC1 Q13547 1/20 0.40
DRD2 P14416 2/20 0.34
IRAK4 Q9NWZ3 1/20 0.33
ENPP2 Q13822 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
ACKR3 P25106 1/20 0.33
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
SIGMAR1 Q99720 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13638887 0.95 S1PR1 (0.47) S1PR1HDAC8HDAC6HDAC1DRD2
SCHEMBL13634595 0.89 S1PR1 (0.49) S1PR1HDAC8HDAC6HDAC1DRD2
SCHEMBL13270598 0.88 S1PR1 (0.41) S1PR1HDAC8HDAC6HDAC1DRD2
SCHEMBL13638884 0.85 S1PR1 (0.47) S1PR1HDAC8HDAC6HDAC1DRD2
SCHEMBL13634748 0.85 S1PR1 (0.36) S1PR1IRAK4CYP1A2CYP3A4CYP2D6
SCHEMBL13634771 0.84 S1PR1 (0.49) S1PR1HDAC8HDAC6HDAC1DRD2
SCHEMBL13162061 0.80 S1PR1 (0.35) S1PR1IRAK4MEN1ALDH1A1CYP1A2
SCHEMBL13634780 0.80 S1PR1 (0.48) S1PR1HDAC8HDAC6HDAC1ENPP2
SCHEMBL13634788 0.80 S1PR1 (0.48) S1PR1HDAC8HDAC6HDAC1DRD2
SCHEMBL13638928 0.80 S1PR1 (0.48) S1PR1HDAC8HDAC6HDAC1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8304547-B2 Azolecarboxamide compound or salt thereof ASTELLAS PHARMA INC. (JP) 2012-11-06 US disclosed