SCHEMBL13639574

SCHEMBL13639574

NC1[C@@H](c2cccc(Cl)c2)[C@H](C(=O)O)N[C@H]1c1cccc(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 2/20 0.38
GRM2 Q14416 1/20 0.36
GRM3 Q14832 1/20 0.36
SLC6A3 Q01959 3/20 0.35
PARP1 P09874 1/20 0.35
HDAC2 Q92769 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
SLC6A2 P23975 1/20 0.34
TP53 P04637 2/20 0.33
MDM2 Q00987 2/20 0.33
ALOX15 P16050 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13639569 0.79 MDM2 (0.39) GRM2GRM3TP53MDM2HTR2A
SCHEMBL13639530 0.79 MDM2 (0.37) SLC9A1GRM2GRM3TP53MDM2
SCHEMBL13639533 0.75 MDM2 (0.49) SLC6A2TP53MDM2
SCHEMBL24737323 0.67 NOTUM (0.40) SLC9A1GRM2GRM3SLC6A3PARP1
SCHEMBL29879161 0.67 NOTUM (0.40) SLC9A1GRM2GRM3SLC6A3PARP1
SCHEMBL29879885 0.65 TRPM4 (0.41) SLC9A1GRM2GRM3SLC6A3TAAR1
SCHEMBL29879030 0.65 TRPM4 (0.41) SLC9A1GRM2GRM3SLC6A3TAAR1
SCHEMBL24737366 0.65 TRPM4 (0.41) SLC9A1GRM2GRM3SLC6A3TAAR1
SCHEMBL21058147 0.65 TP53 (0.48) SLC9A1SLC6A3SLC6A2TP53MDM2
SCHEMBL24378373 0.65 TP53 (0.48) SLC9A1SLC6A3SLC6A2TP53MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2340021-B1 SUBSTITUTED PYRROLIDINE-2-CARBOXAMIDES HOFFMANN LA ROCHE (CH) 2012-11-07 EP disclosed