SCHEMBL13651287

SCHEMBL13651287

COc1cc(N2CCC(=O)[C@@H]2C)ccc1C#N

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AR P10275 12/20 0.52
CHRM4 P08173 1/20 0.38
KCNJ1 P48048 1/20 0.38
KCNH2 Q12809 1/20 0.38
NR3C2 P08235 1/20 0.37
HTR2C P28335 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PKM P14618 1/20 0.36
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13651300 0.82 AR (0.54) AR
SCHEMBL13651229 0.82 AR (0.56) AR
SCHEMBL13651250 0.82 AR (0.56) AR
SCHEMBL13651227 0.79 AR (0.53) AR
SCHEMBL13651289 0.76 AR (0.50) ARCHRM4
SCHEMBL17893756 0.76 AR (0.49) ARCHRM4MEN1KMT2AALDH1A1
SCHEMBL2388777 0.73 AR (0.70) AR
SCHEMBL3339683 0.72 AR (0.55) ARCHRM4NR3C2
SCHEMBL1642826 0.71 AR (0.50) AR
SCHEMBL2390086 0.71 AR (0.47) ARKDM4EUSP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009131196-A1 SUBSTITUTED PYRROLIDINE DERIVATIVE AND USE THEREOF 武田薬品工業株式会社 (JP) 2009-10-29 WO disclosed