SCHEMBL13651289

SCHEMBL13651289

COc1cc(N2CCC[C@@H]2C)ccc1C#N

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.50
ROCK2 O75116 2/20 0.41
ROCK1 Q13464 2/20 0.41
CDC42BPA Q5VT25 2/20 0.41
CDC42BPB Q9Y5S2 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
S1PR1 P21453 1/20 0.41
HTR2A P28223 1/20 0.40
CHRM4 P08173 1/20 0.39
SUV39H2 Q9H5I1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22667722 0.81 AR (0.59) ARROCK2ROCK1CDC42BPACDC42BPB
SCHEMBL13651226 0.81 AR (0.59) ARROCK2ROCK1CDC42BPACDC42BPB
SCHEMBL6236056 0.79 CHRM4 (0.49) MAPTCHRM4
SCHEMBL30664773 0.78 AR (0.49) ARROCK2ROCK1CDC42BPACDC42BPB
SCHEMBL4904736 0.77 AR (0.65) AR
SCHEMBL22667487 0.77 AR (0.65) AR
SCHEMBL13651258 0.77 AR (0.65) AR
SCHEMBL13651287 0.76 AR (0.52) ARCHRM4
SCHEMBL3339683 0.76 AR (0.55) ARCHRM4SUV39H2
SCHEMBL21164657 0.76 ALDH1A1 (0.62) ARMAPTCHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009131196-A1 SUBSTITUTED PYRROLIDINE DERIVATIVE AND USE THEREOF 武田薬品工業株式会社 (JP) 2009-10-29 WO disclosed